(19)
(11) EP 2 643 298 A1

(12)

(43) Date of publication:
02.10.2013 Bulletin 2013/40

(21) Application number: 11788112.8

(22) Date of filing: 21.11.2011
(51) International Patent Classification (IPC): 
C07D 213/61(2006.01)
C07D 213/75(2006.01)
C07D 239/42(2006.01)
C07D 401/12(2006.01)
A61K 31/44(2006.01)
A61P 19/00(2006.01)
A61P 13/12(2006.01)
C07D 213/74(2006.01)
C07D 239/38(2006.01)
C07D 401/04(2006.01)
C07D 403/04(2006.01)
A61K 31/505(2006.01)
A61P 35/00(2006.01)
(86) International application number:
PCT/EP2011/070537
(87) International publication number:
WO 2012/069402 (31.05.2012 Gazette 2012/22)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

(30) Priority: 26.11.2010 US 417369 P

(71) Applicant: Leo Pharma A/S
2750 Ballerup (DK)

(72) Inventors:
  • MÅNSSON, Kristoffer
    DK-2750 Ballerup (DK)
  • BLÆHR, Lars, Kristian, Albert
    DK-2750 Ballerup (DK)

   


(54) SUBSTITUTED CYCLOPENTYL - AZINES AS CASR- ACTIVE COMPOUNDS