(19)
(11) EP 2 685 825 A1

(12)

(43) Date of publication:
22.01.2014 Bulletin 2014/04

(21) Application number: 12757940.7

(22) Date of filing: 14.03.2012
(51) International Patent Classification (IPC): 
A01N 43/42(2006.01)
(86) International application number:
PCT/US2012/029085
(87) International publication number:
WO 2012/125732 (20.09.2012 Gazette 2012/38)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 15.03.2011 US 201161452921 P

(71) Applicant: Vanderbilt University
Nashville, TN 37240 (US)

(72) Inventors:
  • CONN, P., Jeffrey
    Brentwood TN 37027 (US)
  • LINSLEY, Craig, W.
    Brentwood TN 37027 (US)
  • STAUFFER, Shaun, R.
    Brentwood TN 37027 (US)
  • BARTOLOME-NEBREDA, Jose, Manuel
    E-45007 Toledo (ES)
  • MACDONALD, Gregor, James
    2340 Beerse (BE)
  • CONDE-CEIDE, Susana
    E-45007 Toledo (ES)
  • JONES, Carrie, K.
    Nashville TN 37221 (US)
  • MARTIN-MARTIN, Maria, Luz
    E-45007 Toledo (ES)
  • TONG, Han, Min
    E-45007 Toledo (ES)

(74) Representative: Hoefer & Partner 
Pilgersheimer Straße 20
81543 München
81543 München (DE)

   


(54) SUBSTITUTED IMADAZOPYRIMIDIN-5(6H)-ONES AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS