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<ep-patent-document id="EP12725560A1" file="12725560.2" lang="en" country="EP" doc-number="2702043" kind="A1" date-publ="20140305" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRIS..MTNORSMESM..................</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>DIM360 Ver 2.40 (30 Jan 2013) -  1100000/0</B007EP></eptags></B000><B100><B110>2702043</B110><B130>A1</B130><B140><date>20140305</date></B140><B190>EP</B190></B100><B200><B210>12725560.2</B210><B220><date>20120430</date></B220><B240><B241><date>20131030</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201161481035 P</B310><B320><date>20110429</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20140305</date><bnum>201410</bnum></B405><B430><date>20140305</date><bnum>201410</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 239/42        20060101AFI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07D 401/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07D 403/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07D 403/12        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C07D 405/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>C07D 405/12        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>C07D 405/14        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>C07D 409/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>C07D 413/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 417/04        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 417/14        20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="12"><text>A61K  31/506       20060101ALI20121114BHEP        </text></classification-ipcr><classification-ipcr sequence="13"><text>A61P  35/00        20060101ALI20121114BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>INHIBITOREN DER INDUZIERBAREN FORM VON 6-PHOSPHOFRUCTOSE-2-KINASE</B542><B541>en</B541><B542>INHIBITORS OF INDUCIBLE FORM OF 6-PHOSPHOFRUCTOSE-2-KINASE</B542><B541>fr</B541><B542>INHIBITEURS DE LA FORME INDUCTIBLE DE LA 6-PHOSPHOFRUCTOSE-2-KINASE</B542></B540></B500><B700><B710><B711><snm>Exelixis, Inc.</snm><iid>101288191</iid><irf>P162461.EP.01</irf><adr><str>210 East Grand Avenue</str><city>South San Francisco, CA 94080</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>TSUHAKO, Amy, Lew</snm><adr><str>1232 Madruga Way</str><city>Milpitas, CA 95035</city><ctry>US</ctry></adr></B721><B721><snm>MARLOWE, Charles, K.</snm><adr><str>636 California Way</str><city>Emerald Hills, CA 94062</city><ctry>US</ctry></adr></B721><B721><snm>ZAHARIA, Christiana, A.</snm><adr><str>644 Topaz Street</str><city>Redwood City, CA 94061</city><ctry>US</ctry></adr></B721><B721><snm>KABIGTING, Lori</snm><adr><str>349 Commercial Avenue</str><city>South San Francisco, CA 94116</city><ctry>US</ctry></adr></B721><B721><snm>BAJJALIEH, William</snm><adr><str>2086 45th Avenue</str><city>San Francisco, CA 94116</city><ctry>US</ctry></adr></B721><B721><snm>TESFAI, Zerom</snm><adr><str>23219 Canyon Terrace</str><city>Castro Valley, CA 94522</city><ctry>US</ctry></adr></B721><B721><snm>HUANG, Ping</snm><adr><str>117 Whits Road</str><city>Mountain View, CA 94040</city><ctry>US</ctry></adr></B721><B721><snm>MOON, Kim</snm><adr><str>1128 Oregon Avenue</str><city>Palo Alto, CA 94303</city><ctry>US</ctry></adr></B721><B721><snm>AAY, Naing</snm><adr><str>112 N. Rochester Street</str><city>San Mateo, CA 94401</city><ctry>US</ctry></adr></B721><B721><snm>TAMBO-ONG, Arlyn</snm><adr><str>9 N. Spruce Avenue</str><city>South San Francisco, CA 94080</city><ctry>US</ctry></adr></B721><B721><snm>NUSS, John, M.</snm><adr><str>16 Wood Ranch Circle</str><city>Danville, CA 94506</city><ctry>US</ctry></adr></B721><B721><snm>XU, Wei</snm><adr><str>327 Glasgow Circle</str><city>Danville, CA 94526</city><ctry>US</ctry></adr></B721><B721><snm>KEARNEY, Patrick</snm><adr><str>195 Bocana Street</str><city>San Francisco, CA 94110</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Main, Malcolm Charles</snm><iid>100050057</iid><adr><str>Murgitroyd &amp; Company 
Scotland House 
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