PROCESS FOR THE PREPARATION OF PROTEASE INHIBITORS - Patent 2707346

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EP 2 707 346 A1

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(43)	Date of publication:
	19.03.2014 Bulletin 2014/12

(21)	Application number: 12723028.2

(22)	Date of filing: 11.05.2012

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International Patent Classification (IPC):

C07B 53/00^(2006.01)

C07D 209/52^(2006.01)

(86)	International application number:
	PCT/US2012/037515

(87)	International publication number:
	WO 2012/158515 (22.11.2012 Gazette 2012/47)

(84)	Designated Contracting States:
	AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

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Priority:

13.05.2011 US 201161486150 P

(71)	Applicant: Vertex Pharmaceuticals Inc.
	Boston, MA 02210 (US)

(72)	Inventor:
	TANOURY, Gerald, J. Marlborough, MA 01752 (US)

(74)	Representative: Cohausz & Florack
	Patent- und Rechtsanwälte Partnerschaftsgesellschaft Bleichstraße 14 40211 Düsseldorf 40211 Düsseldorf (DE)

(54)	PROCESS FOR THE PREPARATION OF PROTEASE INHIBITORS