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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.63 (23 May 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>2768308</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20180801</date></B140><B150><B151>W1</B151><B153>72</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>12840771.5</B210><B220><date>20121012</date></B220><B240><B241><date>20140513</date></B241><B242><date>20160321</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201161547166 P</B310><B320><date>20111014</date></B320><B330><ctry>US</ctry></B330><B310>201261662163 P</B310><B320><date>20120620</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20180801</date><bnum>201831</bnum></B405><B430><date>20140827</date><bnum>201435</bnum></B430><B450><date>20180418</date><bnum>201816</bnum></B450><B452EP><date>20180308</date></B452EP><B480><date>20180801</date><bnum>201831</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 471/04        20060101AFI20150511BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07H  15/26        20060101ALI20150511BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>C07F   9/6561      20060101ALI20150511BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/47        20060101ALI20150511BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61P  35/00        20060101ALI20150511BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>VERBINDUNGEN UND ANTI-TUMOR-NQO1-SUBSTRATE</B542><B541>en</B541><B542>COMPOUNDS AND ANTI-TUMOR NQO1 SUBSTRATES</B542><B541>fr</B541><B542>COMPOSÉS ET SUBSTRATS ANTITUMORAUX NQO1</B542></B540><B560><B561><text>WO-A2-2012/085532</text></B561><B561><text>US-A- 4 906 562</text></B561><B561><text>US-A- 5 716 963</text></B561><B562><text>PEREZ J M ET AL: "Concise Preparation of 1,8-Diazaanthracene-2,7,9,10-Tetraones. Two Alternative Syntheses of the Natural Antifolate Diazaquinomycin A", TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, vol. 56, no. 26, 1 June 2000 (2000-06-01), pages 4575-4583, XP004202151, ISSN: 0040-4020, DOI: 10.1016/S0040-4020(00)00371-9</text></B562><B562><text>JOSEPH S. BAIR ET AL: "Chemistry and Biology of Deoxynyboquinone, a Potent Inducer of Cancer Cell Death", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. 132, no. 15, 21 April 2010 (2010-04-21), pages 5469-5478, XP055187222, ISSN: 0002-7863, DOI: 10.1021/ja100610m</text></B562><B562><text>X. HUANG ET AL: "An NQO1 Substrate with Potent Antitumor Activity That Selectively Kills by PARP1-Induced Programmed Necrosis", CANCER RESEARCH, vol. 72, no. 12, 15 June 2012 (2012-06-15) , pages 3038-3047, XP055187225, ISSN: 0008-5472, DOI: 10.1158/0008-5472.CAN-11-3135</text></B562><B562><text>DIAZ-GUERRA LUIS M ET AL: "Half-wave potentials of 1-aza and 1,8-diazaanthraquinones", CAPLUS,, 1 January 1995 (1995-01-01), XP002480321,</text></B562><B562><text>LI ET AL.: 'Modulating Endogenous NQ01 Levels Identifies Key Regulatory Mechanisms of Action of b-Lapachone for Pancreatic Cancer Therapy' CLIN CANCER RES vol. 17, no. 2, 15 January 2011, pages 275 - 285, XP055096513</text></B562><B565EP><date>20150518</date></B565EP></B560></B500><B700><B720><B721><snm>HERGENROTHER, Paul J.</snm><adr><str>2607 Wedgewood Drive,</str><city>Champaign, 
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