(19)
(11) EP 2 782 922 A1

(12)

(43) Date of publication:
01.10.2014 Bulletin 2014/40

(21) Application number: 12788225.6

(22) Date of filing: 21.11.2012
(51) International Patent Classification (IPC): 
C07H 17/08(2006.01)
A61P 31/04(2006.01)
 A61K 31/7048(2006.01)
(86) International application number:
PCT/EP2012/073277
(87) International publication number:
WO 2013/076169 (30.05.2013 Gazette 2013/22)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

(30) Priority: 25.11.2011 EP 11190748

(71) Applicants:
  • Bayer Intellectual Property GmbH
    40789 Monheim (DE)
  • The Kitasato Institute
    Tokyo 108-8641 (JP)

(72) Inventors:
  • SATOSHI, Omura
    Setagaya-ku Tokyo 157-0076 (JP)
  • TOSHIAKI, Sunazuka
    Funabashi-shi Chiba 273-0043 (JP)
  • TOMOYASU, Hirose
    Kawasaki-shi Kanagawa 215-0003 (JP)
  • AKIHIRO, Sugawara
    Nerima-ku Tokyo 177-0044 (JP)
  • KAZURO, Shiomi
    Shibuya-ku Tokyo 150-0013 (JP)
  • KLEEFELD, Gerd
    41468 Neuss (DE)
  • FROYMAN, Robrecht
    40789 Monheim (DE)
  • DÖRNER, Julia, Charlotte
    40668 Meerbusch (DE)
  • LUDWIG, Carolin
    40789 Monheim (DE)

(74) Representative: BIP Patents 
c/o Bayer Intellectual Property GmbH Creative Campus Monheim Alfred-Nobel-Straße 10
40789 Monheim
40789 Monheim (DE)

   


(54) ANTIBACTERIAL TYLOSIN DERIVATIVES AND METHODS FOR THEIR PREPARATION