(19)
(11) EP 2 872 500 A2

(12)

(88) Date of publication A3:
06.03.2014

(43) Date of publication:
20.05.2015 Bulletin 2015/21

(21) Application number: 13816563.4

(22) Date of filing: 05.07.2013
(51) International Patent Classification (IPC): 
C07D 401/12(2006.01)
A61P 7/02(2006.01)
A61K 31/4439(2006.01)
(86) International application number:
PCT/IN2013/000413
(87) International publication number:
WO 2014/009966 (16.01.2014 Gazette 2014/03)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 12.07.2012 IN CH28382012
15.10.2012 IN CH42982012

(71) Applicant: Rao, Davuluri Ramamohan
Hyderabad 50003 (IN)

(72) Inventors:
  • PONNAIAH, Ravi
    Madurai 625014 (IN)
  • NEELA, Praveen Kumar
    Hyderabad 500072 (IN)
  • BATTHINI, Guruswamy
    Hyderabad 500082 (IN)
  • VEERA, Narayana B
    Hyderabad 50005 (IN)
  • RAO TELEGAREDDY, Venkata Narasimha
    East Godavari 533247 (IN)
  • BABU, Ravana K
    East Godavari 533445 (IN)

(74) Representative: Dall'Olio, Christian et al
INVENTION S.r.l. Via delle Armi, 1
40137 Bologna
40137 Bologna (IT)

   


(54) AN IMPROVED PROCESS FOR THE PREPARATION OF DABIGATRAN ETEXILATE MESYLATE AND ITS INTERMEDIATES THEREOF