(19)
(11) EP 2 935 254 A1

(12)

(43) Date of publication:
28.10.2015 Bulletin 2015/44

(21) Application number: 13826965.9

(22) Date of filing: 18.12.2013
(51) International Patent Classification (IPC): 
C07D 413/12(2006.01)
A61K 31/537(2006.01)
C07D 498/10(2006.01)
A61K 31/535(2006.01)
C07D 265/22(2006.01)
(86) International application number:
PCT/IB2013/061106
(87) International publication number:
WO 2014/097188 (26.06.2014 Gazette 2014/26)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 21.12.2012 IT MI20122221

(71) Applicant: C4T S.C. a.r.l.
00133 Roma (IT)

(72) Inventors:
  • TOPAI, Alessandra
    I-00133 Roma (IT)
  • MISCIOSCIA, Teresa Fabiola
    I-00133 Roma (IT)
  • BARILE, Fabio
    I-00133 Roma (IT)
  • GUZZO, Tatiana
    I-00133 Roma (IT)
  • MINISSI, Franco
    I-00133 Roma (IT)
  • SABLONE, Manolo
    I-00133 Roma (IT)
  • MACCARRONE, Mauro
    I-00133 Roma (IT)

(74) Representative: Spadaro, Marco et al
Cantaluppi & Partners Via Pellegrino Strobel, 8
20133 Milano
20133 Milano (IT)

   


(54) COMPOUNDS OF 2,3-DIHYDRO-4H-1,3-BENZOXAZINE-4-ONE, METHOD FOR PREPARING THEM AND PHARMACEUTICAL FORM COMPRISING THEM