(19)

(11)

EP 2 935 299 A2

(12)

(88) Date of publication A3: 06.11.2014 (43) Date of publication: 28.10.2015 Bulletin 2015/44 (21) Application number: 13828822.0 (22) Date of filing: 13.12.2013

(51) International Patent Classification (IPC):  C07H 3/06(2006.01) C07K 1/107(2006.01) A61K 47/48(2006.01) A61K 39/09(2006.01) (86) International application number: PCT/IB2013/060933 (87) International publication number: WO 2014/097099 (26.06.2014 Gazette 2014/26)

(84) Designated Contracting States: AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR Designated Extension States: BA ME (30) Priority: 20.12.2012 US 201261740311 P (71) Applicant: Pfizer Inc. New York, NY 10017 (US)	(72) Inventors: HAN, Mingming Nazareth, Pennsylvania 18064 (US) KAINTHAN, Rajesh Kumar Tappan, New York 10983 (US) KIM, Jin-Hwan Suffern, New York 10901 (US) PRASAD, Avvari Krishna Chapel Hill, North Carolina 27516 (US) (74) Representative: Pfizer  European Patent Department 23-25 avenue du Docteur Lannelongue 75668 Paris Cedex 14 75668 Paris Cedex 14 (FR)