(19)
(11) EP 2 956 154 A2

(12)

(88) Date of publication A3:
09.10.2014

(43) Date of publication:
23.12.2015 Bulletin 2015/52

(21) Application number: 14751148.9

(22) Date of filing: 15.02.2014
(51) International Patent Classification (IPC): 
A61K 38/10(2006.01)
(86) International application number:
PCT/US2014/016640
(87) International publication number:
WO 2014/127316 (21.08.2014 Gazette 2014/34)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 15.02.2013 US 201361765423 P
18.06.2013 US 201361836381 P

(71) Applicant: SRX Cardio, LLC
Pittsford, NY 14534 (US)

(72) Inventors:
  • MUEHLEMANN, Michael M.
    Liverpool, NY 13090 (US)
  • BARTA, Thomas E.
    Carrboro, NC 27510 (US)
  • MONROE, Kyle D.
    Pittsford, NY 14534 (US)
  • BOURNE, Jonathan William
    Fairport, NY 14450 (US)
  • REECE, Margaret Thompson
    Fayetteville, NY 13066 (US)
  • NEVALAINEN, Vesa
    Weymouth, MA 02189 (US)

(74) Representative: Grund, Martin 
Grund Intellectual Property Group Postfach 44 05 16
80754 München
80754 München (DE)

   


(54) PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) ALLOSTERIC BINDING LIGANDS TO MUDULATE SERUM LOW DENSITY LIPOPROTEIN (LDL) LEVELS