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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRIS..MTNORSMESM..................</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.63 (23 May 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>2997035</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20180523</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>14723820.8</B210><B220><date>20140514</date></B220><B240><B241><date>20151126</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201361823169 P</B310><B320><date>20130514</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20180523</date><bnum>201821</bnum></B405><B430><date>20160323</date><bnum>201612</bnum></B430><B450><date>20180328</date><bnum>201813</bnum></B450><B452EP><date>20171025</date></B452EP><B480><date>20180523</date><bnum>201821</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07J   9/00        20060101AFI20141127BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>C07J  41/00        20060101ALI20141127BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/575       20060101ALI20141127BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61P   1/16        20060101ALI20141127BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>C07J  71/00        20060101ALI20141127BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>C07J  31/00        20060101ALI20141127BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>11-HYDROXYL-6-SUBSTITUIERTE-DERIVATIVE VON GALLENSÄUREN UND AMINOSÄUREKONJUGATE DAVON ALS FARNESOID-X-REZEPTORMODULATOREN</B542><B541>en</B541><B542>11-HYDROXYL-6-SUBSTITUTED-DERIVATIVES OF BILE ACIDS AND AMINO ACID CONJUGATES THEREOF AS FARNESOID X RECEPTOR MODULATORS</B542><B541>fr</B541><B542>DÉRIVÉS 11-HYDROXYLE D'ACIDES BILIAIRES SUBSTITUÉS EN POSITION 6 ET LEURS CONJUGUÉS D'ACIDES AMINÉS EN TANT QUE MODULATEURS DU RÉCEPTEUR DE FARNÉSOÏDE X</B542></B540><B560><B561><text>EP-A1- 0 124 903</text></B561><B561><text>EP-A1- 1 568 706</text></B561><B561><text>WO-A2-2004/007521</text></B561><B561><text>US-A- 2 802 775</text></B561><B562><text>HITOSHI ISHIDA ET AL: "Study on the Bile Salts from Sunfish, Mola mola L. I. The Structures of Sodium Cyprinol Sulfates, the Sodium Salt of a New Bile Acid Conjugated with Taurine, and a New Bile Alcohol and Its New Sodium Sulfates.", CHEMICAL &amp; PHARMACEUTICAL BULLETIN, vol. 46, no. 1, 1 January 1998 (1998-01-01), pages 12-16, XP55128539, ISSN: 0009-2363, DOI: 10.1248/cpb.46.12</text></B562><B562><text>WILLIAM P LONG ET AL: "PARTIAL SYNTHESIS OF COMPOUNDS RELATED TO ADRENAL CORTICAL HORMONES: III. PREPARATION OF 3([alpha]), 11([alpha])-DIHYDROXYCHOLANIC ACID", J. BIOL. CHEM., vol. 162, no. 3, 1 March 1946 (1946-03-01) , pages 511-519, XP55128534,</text></B562><B562><text>PELLICCIARI R ET AL: "Bile Acid Derivatives as Ligands of the Farnesoid X Receptor. Synthesis, Evaluation, and Structure-Activity Relationship of a Series of Body and Side Chain Modified Analogues of Chenodeoxycholic Acid", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, vol. 47, 23 July 2004 (2004-07-23), pages 4559-4569, XP002370634, ISSN: 0022-2623, DOI: 10.1021/JM049904B</text></B562><B562><text>SIMONA DE MARINO ET AL: "Theonellasterols and Conicasterols from Theonella swinhoei . Novel Marine Natural Ligands for Human Nuclear Receptors", JOURNAL OF MEDICINAL CHEMISTRY, vol. 54, no. 8, 28 April 2011 (2011-04-28) , pages 3065-3075, XP55128555, ISSN: 0022-2623, DOI: 10.1021/jm200169t</text></B562></B560></B500><B600><B620EP><parent><cdoc><dnum><anum>18163622.6</anum></dnum><date>20180323</date></cdoc><cdoc><dnum><anum>18163623.4</anum></dnum><date>20180323</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>PELLICCIARI, Roberto</snm><adr><str>TES Pharma S.r.l.
via Settevalli 556</str><city>I-06129 Perugia</city><ctry>IT</ctry></adr></B721></B720><B730><B731><snm>Intercept Pharmaceuticals, Inc.</snm><iid>101729955</iid><irf>IPHA-020/N01EP</irf><adr><str>10 Hudson Yards, 37th Floor</str><city>New York, NY 10001</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Cooley (UK) LLP</snm><iid>101544956</iid><adr><str>Dashwood 
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