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<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B005EP>J</B005EP><B007EP>BDM Ver 0.1.63 (23 May 2017) -  2999001/0</B007EP></eptags></B000><B100><B110>3002008</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20181024</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>15188438.4</B210><B220><date>20110311</date></B220><B240><B241><date>20160908</date></B241><B242><date>20170111</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>339974 P</B310><B320><date>20100311</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20181024</date><bnum>201843</bnum></B405><B430><date>20160406</date><bnum>201614</bnum></B430><B450><date>20180815</date><bnum>201833</bnum></B450><B452EP><date>20180223</date></B452EP><B480><date>20181024</date><bnum>201843</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  31/535       20060101AFI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/4525      20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/4453      20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/453       20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/5375      20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/495       20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61K  31/496       20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>A61K  31/40        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>A61K  31/404       20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 317/54        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 317/60        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="12"><text>C07D 403/14        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="13"><text>C07D 405/06        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="14"><text>C07C 235/34        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="15"><text>C07C 235/36        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="16"><text>C07D 211/16        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="17"><text>C07D 307/52        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="18"><text>A61P  29/00        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="19"><text>A61P  37/00        20060101ALI20180208BHEP        </text></classification-ipcr><classification-ipcr sequence="20"><text>A61K  31/445       20060101ALI20180208BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>AMIDVERBINDUNGEN ALS RORYT-MODULATOREN UND VERWENDUNGEN DAVON</B542><B541>en</B541><B542>AMIDO COMPOUNDS AS RORYT MODULATORS AND USES THEREOF</B542><B541>fr</B541><B542>COMPOSÉS D'AMIDO COMME MODULATEURS RORYT ET LEURS UTILISATIONS</B542></B540><B560><B561><text>WO-A2-2006/007486</text></B561><B562><text>NARESH KUMAR ET AL: "The Benezenesulfonamide T0901317 [N-(2,2,2-Trifluoroethyl)-N-[4-[2,2,2-trif luoro-1-hydroxy-1-(trifluoromethyl)ethyl]p henyl]-benzenesulfonamide] is a Novel Retinoic Acid Receptor-Related Orphan Receptor-alpha/gamma Inverse Agonist", MOLECULAR PHARMACOLOGY, AMERICAN SOCIETY FOR PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, US, vol. 77, no. 2, 1 February 2010 (2010-02-01), pages 228-236, XP002645391, ISSN: 0026-895X, DOI: 10.1124/MOL.109.060905 [retrieved on 2009-11-03]</text></B562><B562><text>KELIN LI ET AL: "Chemical Libraries via Sequential C-H Functionalization of Phenols", JOURNAL OF COMBINATORIAL CHEMISTRY, vol. 10, no. 2, 1 March 2008 (2008-03-01), pages 170-174, XP055073472, ISSN: 1520-4766, DOI: 10.1021/cc700150q</text></B562><B562><text>Jun R Huh: "Identification of Potent and Selective Diphenylpropanamide ROR[gamma] Inhibitors", ACS Med. Chem. Lett. 2013, 4, 6 December 2012 (2012-12-06), pages 79-84, XP055073467, DOI: 10.1021/ml300286h| Retrieved from the Internet: URL:http://pubs.acs.org/doi/pdf/10.1021/ml 300286h [retrieved on 2013-07-30]</text></B562><B562><text>PASHA M. KHAN ET AL: "Small molecule amides as potent ROR-[gamma] selective modulators", BIOORGANIC &amp; MEDICINAL CHEMISTRY LETTERS, vol. 23, no. 2, 1 January 2013 (2013-01-01), pages 532-536, XP055073469, ISSN: 0960-894X, DOI: 10.1016/j.bmcl.2012.11.025</text></B562></B560></B500><B600><B620><parent><pdoc><dnum><anum>11753726.6</anum><pnum>2558087</pnum></dnum><date>20110311</date></pdoc></parent></B620></B600><B700><B720><B721><snm>Littman, Dan</snm><adr><str>29 Washington Square West
Apartment No. 14D</str><city>New York, NY 1001 1</city><ctry>US</ctry></adr></B721><B721><snm>Huh, Jun, R.</snm><adr><str>435 Riverside Drive No. 81</str><city>New York, NY 10025</city><ctry>US</ctry></adr></B721><B721><snm>Huang, Wenwei</snm><adr><str>317 Oak Knoll Terrace</str><city>Rockville, Maryland</city><ctry>US</ctry></adr></B721><B721><snm>Huang, Ruili</snm><adr><str>514 Jacala Terrace</str><city>Rockville, MD 20850</city><ctry>US</ctry></adr></B721><B721><snm>Englund, Erika, Elaine</snm><adr><str>2900 Connecticut Avenue NW
Apt No. 245</str><city>Washington, DC 20008</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>New York University</snm><iid>101388096</iid><irf>NYU-P1466EPD1</irf><adr><str>70 Washington Square South</str><city>New York, NY 10012</city><ctry>US</ctry></adr></B731><B731><snm>The Government of The United States of America, 
as represented by The Secretary, Department of 
Health and Human Services</snm><iid>101394473</iid><irf>NYU-P1466EPD1</irf><adr><str>National Institutes of Health 
Office of Technology Transfer 
6011 Executive Boulevard, Suite 325</str><city>Rockville, MD 20852-3804</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Teuten, Andrew John</snm><iid>101299088</iid><adr><str>Sagittarius IP 
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