(19)
(11) EP 3 074 389 A1

(12)

(43) Date of publication:
05.10.2016 Bulletin 2016/40

(21) Application number: 13802824.6

(22) Date of filing: 26.11.2013
(51) International Patent Classification (IPC): 
C07D 413/14(2006.01)
A61K 31/517(2006.01)
A61K 35/00(2006.01)
C07D 413/04(2006.01)
A61K 31/4709(2006.01)
(86) International application number:
PCT/US2013/072044
(87) International publication number:
WO 2015/080707 (04.06.2015 Gazette 2015/22)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(71) Applicant: Gilead Sciences, Inc.
Foster City, CA 94404 (US)

(72) Inventors:
  • BABAOGLU, Kerim
    Lansdale, Pennsylvania 19446 (US)
  • CORKEY, Britton Kenneth
    Foster City, California 94404 (US)
  • JIANG, Robert H.
    Cupertino, California 95014 (US)
  • SPERANDIO, David
    Foster City, California 94404 (US)
  • YANG, Hai
    Foster City, California 94404 (US)

(74) Representative: Carpmaels & Ransford LLP 
One Southampton Row
London WC1B 5HA
London WC1B 5HA (GB)

   


(54) QUINOLINE DERIVATIVES AS BROMODOMAIN INHIBITORS