(19)
(11) EP 3 116 873 A1

(12)

(43) Date of publication:
18.01.2017 Bulletin 2017/03

(21) Application number: 15711463.8

(22) Date of filing: 13.03.2015
(51) International Patent Classification (IPC): 
C07D 471/04(2006.01)
A61P 25/00(2006.01)
A61K 31/5513(2006.01)
(86) International application number:
PCT/EP2015/055335
(87) International publication number:
WO 2015/136090 (17.09.2015 Gazette 2015/37)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
MA

(30) Priority: 14.03.2014 US 201461953424 P

(71) Applicant: AbbVie Deutschland GmbH & Co. KG
65189 Wiesbaden (DE)

(72) Inventors:
  • BACKFISCH, Gisela
    67061 Ludwigshafen (DE)
  • BAKKER, Margaretha Henrica Maria
    67061 Ludwigshafen (DE)
  • BLAICH, Günter
    67061 Ludwigshafen (DE)
  • BRAJE, Wilfried
    67061 Ludwigshafen (DE)
  • DRESCHER, Karla
    67061 Ludwigshafen (DE)
  • ERHARD, Thomas
    67061 Ludwigshafen (DE)
  • HAUPT, Andreas
    67061 Ludwigshafen (DE)
  • KOOLMAN, Hannes
    North Chicago, Illinois 60064 (US)
  • LAKICS, Viktor
    67061 Ludwigshafen (DE)
  • REINGRUBER, Anna
    67061 Ludwigshafen (DE)
  • MACK, Helmut
    67061 Ludwigshafen (DE)
  • PETER, Raimund
    Wilmslow SK9 6JB (GB)
  • RELO, Ana Lucia
    67061 Ludwigshafen (DE)
  • WANG, Jincheng
    Tianjin 300457 (CN)
  • ZHAO, Xiaona
    Tianjin 300457 (CN)

(74) Representative: Reitstötter Kinzebach 
Patentanwälte Im Zollhof 1
67061 Ludwigshafen
67061 Ludwigshafen (DE)

   


(54) HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL