(19)
(11) EP 3 119 743 A2

(12)

(88) Date of publication A3:
03.03.2016

(43) Date of publication:
25.01.2017 Bulletin 2017/04

(21) Application number: 14886181.8

(22) Date of filing: 29.12.2014
(51) International Patent Classification (IPC): 
C07C 233/18(2006.01)
(86) International application number:
PCT/IN2014/050008
(87) International publication number:
WO 2015/140812 (24.09.2015 Gazette 2015/38)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME

(30) Priority: 20.03.2014 IN 1492CH2014

(71) Applicant: Biophore India Pharmaceuticals Pvt. Ltd.
Hyderabad 500037 (IN)

(72) Inventors:
  • PULLAGURLA, Manik Reddy
    Hyderabad 500037 (IN)
  • RANGISETTY, Jagadeesh Babu
    Hyderabad 500037 (IN)
  • NANDAKUMAR, Mecheril Valsan
    Hyderabad 500037 (IN)
  • PITTA, Bhaskar Reddy
    Hyderabad 500037 (IN)

(74) Representative: Chas. Hude A/S 
H.C. Andersens Boulevard 33
1780 Copenhagen V
1780 Copenhagen V (DK)

   


(54) AN IMPROVED PROCESS FOR THE PREPARATION OF AGOMELATINE POLYMORPHIC FORM-1