(19)
(11) EP 3 131 880 A1

(12)

(43) Date of publication:
22.02.2017 Bulletin 2017/08

(21) Application number: 15723759.5

(22) Date of filing: 15.04.2015
(51) International Patent Classification (IPC): 
C07D 213/75(2006.01)
C07D 235/12(2006.01)
C07D 405/12(2006.01)
C07D 271/06(2006.01)
C07D 211/44(2006.01)
C07D 213/61(2006.01)
A61K 31/4184(2006.01)
C07D 309/12(2006.01)
C07D 401/12(2006.01)
C07D 471/04(2006.01)
C07D 209/12(2006.01)
C07D 211/46(2006.01)
C07D 305/08(2006.01)
(86) International application number:
PCT/IB2015/052745
(87) International publication number:
WO 2015/159233 (22.10.2015 Gazette 2015/42)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
MA

(30) Priority: 16.04.2014 IN 1379MU2014
22.08.2014 IN 2696MU2014
20.02.2015 IN 545MU2015

(71) Applicant: Glenmark Pharmaceuticals S.A.
2300 La Chaux-de-Fonds (CH)

(72) Inventors:
  • CHAUDHARI, Sachin Sundarlal
    Navi Mumbai Maharashtra 400709 (IN)
  • THOMAS, Abraham
    Navi Mumbai Maharashtra 400705 (IN)
  • KADAM, Ashok Bhausaheb
    Navi Mumbai Maharashtra 400709 (IN)
  • DHONE, Sachin Vasantrao
    Usmanabad Maharashtra 413406 (IN)
  • ADIK, Bharat Gangadhar
    Shrirampur Maharashtra 413739 (IN)
  • KHAIRATKAR-JOSHI, Neelima
    Thane (W) Maharashtra 400602 (IN)
  • SHAH, Daisy Manish
    Mumbai 400028 (IN)
  • BAJPAI, Malini
    Lucknow Uttar Pradesh 226001 (IN)

(74) Representative: HGF Limited 
1 City Walk
Leeds LS11 9DX
Leeds LS11 9DX (GB)

   


(54) ARYL AND HETEROARYL ETHER COMPOUNDS AS ROR GAMMA MODULATORS