(19)
(11) EP 3 197 875 A1

(12)

(43) Date of publication:
02.08.2017 Bulletin 2017/31

(21) Application number: 15782120.8

(22) Date of filing: 25.09.2015
(51) International Patent Classification (IPC): 
C07D 239/70(2006.01)
(86) International application number:
PCT/US2015/052143
(87) International publication number:
WO 2016/049414 (31.03.2016 Gazette 2016/13)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
MA

(30) Priority: 26.09.2014 US 201462055893 P

(71) Applicants:
  • F. Hoffmann-La Roche AG
    4070 Basel (CH)
  • Genentech, Inc.
    South San Francisco, CA 94080-4990 (US)

(72) Inventors:
  • GOSSELIN, Francis
    South San Francisco, California 94080-4990 (US)
  • HAN, Chong
    South San Francisco, California 94080-4990 (US)
  • IDING, Hans
    CH-4070 Basel (CH)
  • REENTS, Reinhard
    CH-4070 Basel (CH)
  • SAVAGE, Scott
    South San Francisco, California 94080-4990 (US)
  • WIRZ, Beat
    CH-4070 Basel (CH)

(74) Representative: Bailey, Sam Rogerson et al
Mewburn Ellis LLP City Tower 40 Basinghall Street
London EC2V 5DE
London EC2V 5DE (GB)

   


(54) PROCESSES FOR PREPARING (CYCLOPENTYL[d]PYRIMIDIN-4-YL)PIPERAZINE COMPOUNDS