(19)
(11) EP 3 202 404 A8

(12) CORRECTED EUROPEAN PATENT APPLICATION
published in accordance with Art. 153(4) EPC

(15) Correction information:
Corrected version no 1 (W1 A1)

(48) Corrigendum issued on:
14.02.2018 Bulletin 2018/07

(43) Date of publication:
09.08.2017 Bulletin 2017/32

(21) Application number: 15847156.5

(22) Date of filing: 28.09.2015
(51) International Patent Classification (IPC): 
A61K 31/569(2006.01)
A61K 47/30(2006.01)
A61K 47/14(2017.01)
A61P 13/08(2006.01)
A61K 9/00(2006.01)
A61K 47/38(2006.01)
A61K 47/26(2006.01)
A61P 35/00(2006.01)
A61K 9/20(2006.01)
(86) International application number:
PCT/CN2015/090951
(87) International publication number:
WO 2016/050193 (07.04.2016 Gazette 2016/14)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

(30) Priority: 29.09.2014 CN 201410520235

(71) Applicant: Chen, Yajun
Shanghai 200002 (CN)

(72) Inventor:
  • Chen, Yajun
    Shanghai 200002 (CN)

(74) Representative: Di Giovine, Paolo et al
Società Italiana Brevetti S.p.A. Piazza di Pietra, 38-39
00186 Roma
00186 Roma (IT)


(56) References cited: : 
   
       


    (54) ORAL FORMULATION OF A-NOR-5ALPHA ANDROSTANE COMPOUND


    (57) An oral formulation, and preparation method and use thereof; the oral formulation comprises 1-50 parts by weight of an A-nor-5α-androstane compound, 20-95 parts by weight of a filling agent, 0-20 parts by weight of a disintegrant, 0.1-30 parts by weight of a binder, 0.1-5 parts by weight of a lubricant and 0.1-5 parts by weight of a glidant. The oral formulation has a high stability and a good dissolution performance.