ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................*JBDM Ver 2.0.14 (4th of August) - 2999001/03307251CORRECTED EUROPEAN PATENT SPECIFICATIONB8B120211201W173deBibliographieenBibliographyfrBibliographieEP16730210.8201606092018010820191112enenen201562173174 P20150609US201562210708 P20150827US201662289801 P20160201US201662319369 P20160407US2021120120214820180418201816202110202021422021012620211201202148C07D 239/47 20060101AFI20201221BHEP C07D 201/00 20060101ALI20201221BHEP C07K 16/00 20060101ALI20201221BHEP A61K 31/513 20130101 LI20160719BHEP A61K2300/00 20130101 LI20160719BHEP C12Y 207/01048 20130101 LI20170119BHEP A61P 35/00 20180101 LI20200327BHEP A61K 9/2004 20130101 LA20170626BHEP C07D 239/47 20130101 LI20160719BHEP A61K 31/513 20130101 FI20160719BHEP G01N2800/52 20130101 LA20170802BHEP A61K 9/4841 20130101 LA20170626BHEP A61K2039/505 20130101 LA20170119BHEP deFLUOROCYCLOPENTENYLCYTOSIN, VERWENDUNG UND VERFAHREN ZUR HERSTELLUNGenFLUOROCYCLOPENTENYLCYTOSINE USES AND PROCESSES OF PREPARATIONfrUTILISATIONS DE FLUOROCYCLOPENTÉNYLCYTOSINE ET PROCÉDÉS DE PRÉPARATION DE CE COMPOSÉWO-A2-2005/097757US-A1- 2014 275 537Mi Young Yang ET AL: "A novel cytidine analog, RX-3117, shows potent efficacy in xenograft models, even in tumors that are resistant to gemcitabine", Anticancer research, December 2014 (2014-12), page 6951, XP055289638, Greece Retrieved from the Internet: URL:http://ar.iiarjournals.org/content/34/ 12/6951.full.pdf [retrieved on 2016-07-22] cited in the applicationWON JUN CHOI ET AL: "Fluorocyclopentenyl-cytosine with Broad Spectrum and Potent Antitumor Activity +", JOURNAL OF MEDICINAL CHEMISTRY, vol. 55, no. 9, 10 May 2012 (2012-05-10), pages 4521-4525, XP055120207, ISSN: 0022-2623, DOI: 10.1021/jm3004009 cited in the applicationISTVAN UDVAROS ET AL: "A phase 1 exploratory study of RX-3117 to determine oral bioavailability in cancer subjects with solid tumors.", JOURNAL OF CLINICAL ONCOLOGY, vol. 33, no. 15 (suppl), 20 May 2015 (2015-05-20), page e13545, XP055290526,21203072.020211018LEE, Young Bok15245 Shady Grove Road Suite 455Rockville, Maryland 20850USKIM, Deog Joong15245 Shady Grove Road Suite 455Rockville, Maryland 20850USPETERS, Godefridus J.Department of Medical Oncology VU University Medical Center P.O. Box 70571007 MB AmsterdamNLSARKISJAN, Dzjemma40 allée du mail92360 MeudonFRMAZHARI, Reza15245 Shady Grove Road Suite 455Rockville, Maryland 20850USOcuphire Pharma, Inc.101922189172547EP CS/vg15245 Shady Grove Road, Suite 455Rockville, MD 20850USdompatent von Kreisler Selting Werner - Partnerschaft von Patent- und Rechtsanwälten mbB101166970Deichmannhaus am Dom Bahnhofsvorplatz 150667 KölnDEALATBEBGCHCYCZDEDKEEESFIFRGBGRHRHUIEISITLILTLULVMCMKMTNLNOPLPTRORSSESISKSMTRUS201603676820160609enWO201620114620161215201650