<?xml version="1.0" encoding="UTF-8"?>
<!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.5.1//EN" "ep-patent-document-v1-5-1.dtd">
<!-- This XML data has been generated under the supervision of the European Patent Office -->
<ep-patent-document id="EP16734529B8W1" file="EP16734529W1B8.xml" lang="en" country="EP" doc-number="3310760" kind="B8" correction-code="W1" date-publ="20221019" status="c" dtd-version="ep-patent-document-v1-5-1">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRIS..MTNORSMESMMA....MD..........</B001EP><B003EP>*</B003EP><B005EP>J</B005EP><B007EP>BDM Ver 2.0.16 (1th of February 2022) -  2999001/0</B007EP></eptags></B000><B100><B110>3310760</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20221019</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>16734529.7</B210><B220><date>20160621</date></B220><B240><B241><date>20180117</date></B241><B242><date>20181220</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201562182841 P</B310><B320><date>20150622</date></B320><B330><ctry>US</ctry></B330><B310>201562207531 P</B310><B320><date>20150820</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20221019</date><bnum>202242</bnum></B405><B430><date>20180425</date><bnum>201817</bnum></B430><B450><date>20220914</date><bnum>202237</bnum></B450><B452EP><date>20220504</date></B452EP><B480><date>20221019</date><bnum>202242</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 209/94        20060101AFI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/403       20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61P  37/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>A61P  29/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="5"><text>A61P  35/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="6"><text>A61P   9/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P   1/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="8"><text>A61P   7/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="9"><text>A61P   3/00        20060101ALI20170112BHEP        </text></classification-ipcr><classification-ipcr sequence="10"><text>A61P   5/00        20060101ALI20170112BHEP        </text></classification-ipcr></B510EP><B520EP><classifications-cpc><classification-cpc sequence="1"><text>C07D 209/94        20130101 FI20160727BHEP        </text></classification-cpc><classification-cpc sequence="2"><text>A61P   1/00        20180101 LI20200318BHEP        </text></classification-cpc><classification-cpc sequence="3"><text>A61P   1/04        20180101 LI20200318BHEP        </text></classification-cpc><classification-cpc sequence="4"><text>A61P   1/16        20180101 LI20200318BHEP        </text></classification-cpc><classification-cpc sequence="5"><text>A61P  17/02        20180101 LI20200319BHEP        </text></classification-cpc><classification-cpc sequence="6"><text>A61P  17/06        20180101 LI20200320BHEP        </text></classification-cpc><classification-cpc sequence="7"><text>A61P  17/10        20180101 LI20200320BHEP        </text></classification-cpc><classification-cpc sequence="8"><text>A61P  19/02        20180101 LI20200320BHEP        </text></classification-cpc><classification-cpc sequence="9"><text>A61P  25/00        20180101 LI20200320BHEP        </text></classification-cpc><classification-cpc sequence="10"><text>A61P  29/00        20180101 LI20200324BHEP        </text></classification-cpc><classification-cpc sequence="11"><text>A61P   3/00        20180101 LI20200326BHEP        </text></classification-cpc><classification-cpc sequence="12"><text>A61P  35/00        20180101 LI20200327BHEP        </text></classification-cpc><classification-cpc sequence="13"><text>A61P  37/00        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="14"><text>A61P  37/02        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="15"><text>A61P  43/00        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="16"><text>A61P   5/00        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="17"><text>A61P   7/00        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="18"><text>A61P   9/00        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="19"><text>A61P   3/10        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="20"><text>C07C 279/14        20130101 LI20210922BHEP        </text></classification-cpc></classifications-cpc></B520EP><B540><B541>de</B541><B542>KRISTALLINES L-ARGININSALZ VON (R) -2-(7-(4-CYCLOPENTYL-3-(TRIFLUORMETHYL) BENZYLOXY ) -1,2,3,4-TETRAHYDROCYCLO-PENTA [ B ] INDOL-3-YL) ESSIGSÄURE ZUR VERWENDUNG BEI S1P1-REZEPTOR-ASSOZIERTEN ERKRANKUNGEN</B542><B541>en</B541><B542>CRYSTALLINE  L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3,4-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACETIC ACID FOR USE IN S1P1 RECEPTOR-ASSOCIATED DISORDERS</B542><B541>fr</B541><B542>SEL L-ARGININE CRISTALLIN D'ACIDE (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMÉTHYL)BENZYLOXY)-1,2,3,4-TÉTRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACÉTIQUE POUR UNE UTILISATION DANS DES TROUBLES ASSOCIÉS AU RÉCEPTEUR DE S1P1</B542></B540><B560><B561><text>WO-A1-2010/011316</text></B561><B561><text>WO-A1-2011/094008</text></B561><B562><text>NORBERT RASENACK ET AL: "Crystal habit and tableting behavior", INTERNATIONAL JOURNAL OF PHARMACEUTICS, vol. 244, no. 1-2, 1 September 2002 (2002-09-01), pages 45-57, XP055291502, NL ISSN: 0378-5173, DOI: 10.1016/S0378-5173(02)00296-X</text></B562></B560></B500><B600><B620EP><parent><cdoc><dnum><anum>21178613.2</anum><pnum>3939965</pnum></dnum><date>20210609</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>BLACKBURN, Anthony C.</snm><adr><str>12633 Caminito Rosita</str><city>San Diego, California 92128</city><ctry>US</ctry></adr></B721><B721><snm>CASTRO, Ryan O.</snm><adr><str>8706 Elford Court</str><city>San Diego, California 92129</city><ctry>US</ctry></adr></B721><B721><snm>HADD, Mark A.</snm><adr><str>8544 Ivory Coast Drive</str><city>San Diego, California 92126</city><ctry>US</ctry></adr></B721><B721><snm>MA, You-An</snm><adr><str>12820 Oakfield Way</str><city>Poway, California 92064</city><ctry>US</ctry></adr></B721><B721><snm>MONTALBAN, Antonio Garrido</snm><adr><str>10339 Azuaga Street
No. 213</str><city>San Diego, California 92129</city><ctry>US</ctry></adr></B721><B721><snm>RUETER, Jaimie Karyn</snm><adr><str>9022 Westvale Road</str><city>San Diego, California 92129</city><ctry>US</ctry></adr></B721><B721><snm>SELVEY, Lee Alani</snm><adr><str>12976 Cree Drive</str><city>Poway, California 92064</city><ctry>US</ctry></adr></B721><B721><snm>SHAKYA, Sagar Raj</snm><adr><str>12180 Dormouse Road</str><city>San Diego, California 92129</city><ctry>US</ctry></adr></B721><B721><snm>CARLOS, Marlon</snm><adr><str>1414 Klamath Drive</str><city>Chula Vista, California 91913</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>Arena Pharmaceuticals, Inc.</snm><iid>101962549</iid><irf>007326655</irf><adr><str>235 East 42nd Street</str><city>New York, NY 10017</city><ctry>US</ctry></adr></B731></B730><B740><B741><snm>Mewburn Ellis LLP</snm><iid>101783151</iid><adr><str>Aurora Building 
Counterslip</str><city>Bristol BS1 6BX</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AL</ctry><ctry>AT</ctry><ctry>BE</ctry><ctry>BG</ctry><ctry>CH</ctry><ctry>CY</ctry><ctry>CZ</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>EE</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>HR</ctry><ctry>HU</ctry><ctry>IE</ctry><ctry>IS</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LT</ctry><ctry>LU</ctry><ctry>LV</ctry><ctry>MC</ctry><ctry>MK</ctry><ctry>MT</ctry><ctry>NL</ctry><ctry>NO</ctry><ctry>PL</ctry><ctry>PT</ctry><ctry>RO</ctry><ctry>RS</ctry><ctry>SE</ctry><ctry>SI</ctry><ctry>SK</ctry><ctry>SM</ctry><ctry>TR</ctry></B840><B844EP><B845EP><ctry>BA</ctry><date>20180117</date></B845EP><B845EP><ctry>ME</ctry><date>20180117</date></B845EP></B844EP><B848EP><B849EP><ctry>MA</ctry><date>20180117</date></B849EP><B849EP><ctry>MD</ctry><date>20180117</date></B849EP></B848EP><B860><B861><dnum><anum>US2016038506</anum></dnum><date>20160621</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO2016209809</pnum></dnum><date>20161229</date><bnum>201652</bnum></B871></B870></B800></SDOBI>
</ep-patent-document>
