(19)
(11) EP 3 487 854 A1

(12)

(43) Date of publication:
29.05.2019 Bulletin 2019/22

(21) Application number: 17740021.5

(22) Date of filing: 17.07.2017
(51) International Patent Classification (IPC): 
C07D 409/12(2006.01)
C07D 215/14(2006.01)
C07D 409/14(2006.01)
(86) International application number:
PCT/EP2017/068058
(87) International publication number:
WO 2018/015354 (25.01.2018 Gazette 2018/04)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
MA MD

(30) Priority: 19.07.2016 PL 41801916

(71) Applicant: Adamed Pharma S.A.
05-152 Czosnow (PL)

(72) Inventors:
  • RUSIECKI, Rafal
    01-891 Warszawa (PL)
  • SNIEZEK, Marcin
    03-287 Warszawa (PL)

(74) Representative: Sulikowski, Daniel 
Admarka sp. z o.o. Pienków, ul. Mariana Adamkiewicza 6
05-152 Czosnów
05-152 Czosnów (PL)

   


(54) THE METHOD FOR MANUFACTURE OF BREXPIPRAZOLE, INTERMEDIATES USED IN THIS METHOD, AND THE METHOD FOR MANUFACTURE THEREOF