(19)
(11) EP 3 493 814 A1

(12)

(43) Date of publication:
12.06.2019 Bulletin 2019/24

(21) Application number: 17837574.7

(22) Date of filing: 01.08.2017
(51) International Patent Classification (IPC): 
A61K 31/66(2006.01)
C07F 9/02(2006.01)
(86) International application number:
PCT/US2017/044984
(87) International publication number:
WO 2018/026866 (08.02.2018 Gazette 2018/06)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
MA MD

(30) Priority: 03.08.2016 US 201662370637 P

(71) Applicant: Neuropore Therapies, Inc.
San Diego, CA 92121 (US)

(72) Inventors:
  • WRASIDLO, Wolfgang
    San Diego CA 92121 (US)
  • NATALA, Srinivasa, Reddy
    San Diego CA 92121 (US)

(74) Representative: Mewburn Ellis LLP 
City Tower 40 Basinghall Street
London EC2V 5DE
London EC2V 5DE (GB)

   


(54) LIPID-SUBSTITUTED AMINO 1,2-AND 1,3-DIOL COMPOUNDS AS MODULATORS OF TLR2 DIMERIZATION