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<ep-patent-document id="EP18152422B8W1" file="EP18152422W1B8.xml" lang="de" country="EP" doc-number="3514235" kind="B8" correction-code="W1" date-publ="20240214" status="c" dtd-version="ep-patent-document-v1-6">
<SDOBI lang="de"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSK..HRIS..MTNORS..SM..................</B001EP><B005EP>J</B005EP><B007EP>BDM Ver 2.0.24 -  2999001/0</B007EP></eptags></B000><B100><B110>3514235</B110><B120><B121>KORRIGIERTE EUROPÄISCHE PATENTSCHRIFT</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20240214</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>18152422.4</B210><B220><date>20180118</date></B220><B240><B241><date>20200124</date></B241><B242><date>20200221</date></B242></B240><B250>de</B250><B251EP>de</B251EP><B260>de</B260></B200><B400><B405><date>20240214</date><bnum>202407</bnum></B405><B430><date>20190724</date><bnum>201930</bnum></B430><B450><date>20240103</date><bnum>202401</bnum></B450><B452EP><date>20231025</date></B452EP><B480><date>20240214</date><bnum>202407</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C12N  15/113       20100101AFI20180530BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/7088      20060101ALI20180530BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61P   1/00        20060101ALI20180530BHEP        </text></classification-ipcr></B510EP><B520EP><classifications-cpc><classification-cpc sequence="1"><text>C12N  15/113       20130101 FI20180518BHEP        </text></classification-cpc><classification-cpc sequence="2"><text>C12N  15/1136      20130101 LI20180518BHEP        </text></classification-cpc><classification-cpc sequence="3"><text>C12N2310/127       20130101 LA20180518BHEP        </text></classification-cpc></classifications-cpc></B520EP><B540><B541>de</B541><B542>ZUSAMMENSETZUNG ZUR BEHANDLUNG EINES AN COLITIS ULCEROSA LEIDENDEN PATIENTEN SOWIE VERWENDUNG DER ZUSAMMENSETZUNG ALS ARZNEIMITTEL</B542><B541>en</B541><B542>COMPOSITION FOR THE TREATMENT OF A PATIENT SUFFERING FROM ULCERATIVE COLITIS AND UTILISATION OF SAID COMPOSITION AS MEDICAMENT</B542><B541>fr</B541><B542>COMPOSITION DESTINÉE AU TRAITEMENT DE PATIENTS SOUFFRANT D'UNE COLITE ULCEREUSE AINSI QUE L'UTILISATION DE LADITE COMPOSITION EN TANT QUE MÉDICAMENT</B542></B540><B560><B561><text>WO-A1-2017/205506</text></B561><B561><text>WO-A2-2005/033314</text></B561><B561><text>WO-A2-2014/040891</text></B561><B561><text>US-A1- 2003 040 497</text></B561><B562><text>POPP VANESSA ET AL: "Rectal Delivery of a DNAzyme That Specifically Blocks the Transcription Factor GATA3 and Reduces Colitis in Mice", GASTROENTEROLOGY, W.B. SAUNDERS CO, US, Bd. 152, Nr. 1, 14. September 2016 (2016-09-14), Seiten 176-192, XP029851140, ISSN: 0016-5085, DOI: 10.1053/J.GASTRO.2016.09.005</text></B562><B562><text>Anonymous: "DRKS-ID: DRKS00007193 SB012 for the Treatment of Active Ulcerative Colitis (SECURE): a Prospective, Single-centre, Randomised, Double-blind, Placebo-controlled Phase IIa Clinical Trial to Evaluate the Efficacy, Pharmacokinetics, Tolerability, and Safety of SB012 Enema Administered Once Daily", , 9. Juni 2015 (2015-06-09), XP055476967, Gefunden im Internet: URL:http://www.drks.de/drks_web/navigate.d o?navigationId=trial.HTML&amp;TRIAL_ID=DRKS000 07193 [gefunden am 2018-05-18]</text></B562><B562><text>WEIGMANN BENNO ET AL: "Suppression of Experimental Ulcerative Colitis by Topical Delivery of Specific Dnazyme Blocking Thetranscription Factor GATA3", GASTROENTEROLOGY, W.B. SAUNDERS CO, US, 22. April 2017 (2017-04-22), XP085104521, ISSN: 0016-5085, DOI: 10.1016/S0016-5085(17)32631-8</text></B562><B562><text>KATRINA RAY: "A role for GATA3 in ulcerative colitis", NATURE REVIEWS / GASTROENTEROLOGY &amp; HEPATOLOGY, Bd. 13, Nr. 11, 5. Oktober 2016 (2016-10-05), Seiten 624-624, XP55476486, US ISSN: 1759-5045, DOI: 10.1038/nrgastro.2016.163</text></B562><B562><text>ALESYA A. FOKINA ET AL: "Delivery of therapeutic RNA-cleaving oligodeoxyribonucleotides (deoxyribozymes): from cell culture studies to clinical trials", EXPERT OPINION ON DRUG DELIVERY, Bd. 14, Nr. 9, 7. Dezember 2016 (2016-12-07), Seiten 1077-1089, XP55476495, GB ISSN: 1742-5247, DOI: 10.1080/17425247.2017.1266326</text></B562><B562><text>URBANSKA ALEKSANDRA M ET AL: "What's Next for Gastrointestinal Disorders: No Needles?", JOURNAL OF CONTROLLED RELEASE, Bd. 221, 2. Dezember 2015 (2015-12-02), Seiten 48-61, XP029383249, ISSN: 0168-3659, DOI: 10.1016/J.JCONREL.2015.11.031</text></B562><B562><text>Zhijie Xu ET AL: "Small-molecule Nucleic-acid-based Gene-silencing Strategies" In: "Nucleic Acids - From Basic Aspects to Laboratory Tools", 16. März 2016 (2016-03-16), InTech, XP55476951, ISBN: 978-953-51-2264-7 DOI: 10.5772/62137, * Tabelle 2 *</text></B562><B562><text>HOLGER GARN ET AL: "GATA-3-specific DNAzyme - A novel approach for stratified asthma therapy", EUROPEAN JOURNAL OF IMMUNOLOGY, Bd. 47, Nr. 1, 2. Dezember 2016 (2016-12-02), Seiten 22-30, XP055476945, ISSN: 0014-2980, DOI: 10.1002/eji.201646450</text></B562><B562><text>COMINELLI FABIO ET AL: "Uncovering Pathogenic Mechanisms of Inflammatory Bowel Disease Using Mouse Models of Crohn's Disease-Like Ileitis: What is the Right Model?", CELLULAR AND MOLECULAR GASTROENTEROLOGY AND HEPATOLOGY JUL 2017, vol. 4, no. 1, July 2017 (2017-07), pages 19-32, ISSN: 2352-345X</text></B562><B562><text>KOELINK PJ AND TE VELDE AA: "Mistakes in mouse models of IBD and how to avoid them.", UEG EDUCATION, vol. 16, 2016, pages 11-14,</text></B562><B562><text>NGUYEN THI LOAN ANH ET AL: "How informative is the mouse for human gut microbiota research?", DISEASE MODELS &amp; MECHANISMS JAN 2015, vol. 8, no. 1, January 2015 (2015-01), pages 1-16, ISSN: 1754-8411</text></B562><B562><text>ALDARS-GARCÍA LAILA ET AL: "The Interplay between Immune System and Microbiota in Inflammatory Bowel Disease: A Narrative Review.", INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES 17 MAR 2021, vol. 22, no. 6, 17 March 2021 (2021-03-17) , ISSN: 1422-0067</text></B562><B562><text>CROUWEL FEMKE ET AL: "Gut microbiota-driven drug metabolism in inflammatory bowel disease.", JOURNAL OF CROHN'S &amp; COLITIS 11 JUL 2020, 11 July 2020 (2020-07-11), ISSN: 1876-4479</text></B562><B562><text>VALATAS VASSILIS ET AL: "The value of experimental models of colitis in predicting efficacy of biological therapies for inflammatory bowel diseases.", AMERICAN JOURNAL OF PHYSIOLOGY. GASTROINTESTINAL AND LIVER PHYSIOLOGY DEC 2013, vol. 305, no. 11, December 2013 (2013-12), pages G763-G785, ISSN: 1522-1547</text></B562><B562><text>VICTOR JULIAN ET AL: "Inability of DNAzymes to cleave RNA in vivo is due to limited Mg[Formula: see text] concentration in cells.", EUROPEAN BIOPHYSICS JOURNAL : EBJ MAY 2018, vol. 47, no. 4, May 2018 (2018-05), pages 333-343, ISSN: 1432-1017</text></B562><B562><text>TRAPANI VALENTINA ET AL: "Dietary Magnesium Alleviates Experimental Murine Colitis Through Upregulation of the Transient Receptor Potential Melastatin 6 Channel.", INFLAMMATORY BOWEL DISEASES 15 09 2018, vol. 24, no. 10, 15 September 2018 (2018-09-15), pages 2198-2210, ISSN: 1536-4844</text></B562><B562><text>SWANSON KENNETH D ET AL: "Reproducing the human mucosal environment ex vivo: inflammatory bowel disease as a paradigm.", CURRENT OPINION IN GASTROENTEROLOGY 11 2018, vol. 34, no. 6, November 2018 (2018-11), pages 384-391, ISSN: 1531-7056</text></B562></B560></B500><B700><B720><B721><snm>Renz, Jonas</snm><adr><str>Höchlstr. 3</str><city>81675 München</city><ctry>DE</ctry></adr></B721></B720><B730><B731><snm>Sterna Biologicals GmbH</snm><iid>102025158</iid><irf>SCR19P02EP1</irf><adr><str>Rudolf-Bultmann-Str. 4h</str><city>35039 Marburg</city><ctry>DE</ctry></adr></B731></B730><B740><B741><snm>Pharma Patents International AG</snm><iid>101562763</iid><adr><str>Leonhardsgraben 52 
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