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<ep-patent-document id="EP17888222A1" file="17888222.1" lang="en" country="EP" doc-number="3565600" kind="A1" date-publ="20191113" status="n" dtd-version="ep-patent-document-v1-5"><!-- This XML data has been generated under the supervision of the European Patent Office --><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRIS..MTNORSMESMMA..TNMD..........</B001EP><B003EP>*</B003EP><B005EP>X</B005EP><B007EP>BDM Ver 0.1.67 (18 Oct 2017) -  1100000/0</B007EP></eptags></B000><B100><B110>3565600</B110><B130>A1</B130><B140><date>20191113</date></B140><B190>EP</B190></B100><B200><B210>17888222.1</B210><B220><date>20171228</date></B220><B240><B241><date>20190528</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201662440658 P</B310><B320><date>20161230</date></B320><B330><ctry>US</ctry></B330><B310>PCT/US2017/039968</B310><B320><date>20170629</date></B320><B330><ctry>WO</ctry></B330><B310>201715637401</B310><B320><date>20170629</date></B320><B330><ctry>US</ctry></B330><B310>2972296</B310><B320><date>20170629</date></B320><B330><ctry>CA</ctry></B330></B300><B400><B405><date>20191113</date><bnum>201946</bnum></B405><B430><date>20191113</date><bnum>201946</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  47/10        20170101AFI20180706BHEP        </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  47/14        20170101ALI20180706BHEP        </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  47/26        20060101ALI20180706BHEP        </text></classification-ipcr><classification-ipcr sequence="4"><text>C07C  31/08        20060101ALI20180706BHEP        </text></classification-ipcr></B510EP><B540><B541>de</B541><B542>DEPOTFORMULIERUNGEN</B542><B541>en</B541><B542>DEPOT FORMULATIONS</B542><B541>fr</B541><B542>PRÉPARATIONS DÉPÔT</B542></B540></B500><B700><B710><B711><snm>Durect Corporation</snm><iid>101726298</iid><irf>N416798EP</irf><adr><str>10260 Bubb Road</str><city>Cupertino, CA 95014-4166</city><ctry>US</ctry></adr></B711><B711><snm>Santen Pharmaceutical Co., Ltd.</snm><iid>101581750</iid><irf>N416798EP</irf><adr><str>9-19, Shimoshinjo 3-chome</str><city>Higashiyodogawa-ku
Osaka-shi
Osaka 533-8651</city><ctry>JP</ctry></adr></B711></B710><B720><B721><snm>TAMRAZ, Wilma</snm><adr><str>7002 Noonwood Ct.</str><city>San Jose
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California 95120</city><ctry>US</ctry></adr></B721><B721><snm>LIN, WeiQi</snm><adr><str>590 California Way</str><city>Emerald Hills
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8916-16 Takayama-cho</str><city>Ikoma-shi
Nara 630-0101</city><ctry>JP</ctry></adr></B721><B721><snm>MATSUMOTO, Naoki</snm><adr><str>c/o SANTEN PHARMACEUTICAL CO. LTD.
8916-16 Takayama-cho</str><city>Ikoma-shi
Nara 630-0101</city><ctry>JP</ctry></adr></B721><B721><snm>MUDUMBA, Sreenivasu</snm><adr><str>c/o Santen Inc.
2100 Powell Street
Suite 1600</str><city>Emeryville
California 94608</city><ctry>US</ctry></adr></B721><B721><snm>OKABE, Komei</snm><adr><str>c/o Santen Pharmaceutical Co. Ltd.
8916-16 Takayama-cho</str><city>Ikoma-shi
Nara 630-0101</city><ctry>JP</ctry></adr></B721></B720><B740><B741><snm>J A Kemp LLP</snm><iid>101669666</iid><adr><str>14 South Square 
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