(19)
(11) EP 3 630 778 A1

(12)

(43) Date of publication:
08.04.2020 Bulletin 2020/15

(21) Application number: 18728587.9

(22) Date of filing: 28.05.2018
(51) International Patent Classification (IPC): 
C07D 498/04(2006.01)
A61K 31/519(2006.01)
A61K 31/4375(2006.01)
A61P 35/00(2006.01)
(86) International application number:
PCT/EP2018/063957
(87) International publication number:
WO 2018/215668 (29.11.2018 Gazette 2018/48)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 26.05.2017 US 201762511455 P
11.08.2017 US 201762544531 P

(71) Applicant: Ichnos Sciences SA
2300 La Chaux-de-Fonds (CH)

(72) Inventors:
  • PATEL, Vinod
    2300 La Chaux-de-Fonds (CH)
  • REDDY, Venkateshwar
    2300 La Chaux-de-Fonds (CH)
  • GHARAT, Laxmikant Atmaram
    2300 La Chaux-de-Fonds (CH)
  • CHAUDHARI, Sachin Sundarlal
    2300 La Chaux-de-Fonds (CH)
  • DAS, Sanjib
    2300 La Chaux-de-Fonds (CH)
  • VELGALETI, Ranganadh
    2300 La Chaux-de-Fonds (CH)
  • SHAH, Daisy Manish
    2300 La Chuax-de-Fonds (CH)
  • BAJPAI, Malini
    2300 La Chaux-de-Fonds (CH)

   


(54) NOVEL INHIBITORS OF MAP4K1