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<ep-patent-document id="EP20153723B8W1" file="EP20153723W1B8.xml" lang="en" country="EP" doc-number="3715345" kind="B8" correction-code="W1" date-publ="20240529" status="c" dtd-version="ep-patent-document-v1-6">
<SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIESILTLVFIROMKCYALTRBGCZEEHUPLSKBAHRIS..MTNORSMESM..................</B001EP><B005EP>J</B005EP><B007EP>BDM Ver 2.0.26 -  2999001/0</B007EP><B070EP>The file contains technical information submitted after the application was filed and not included in this specification</B070EP></eptags></B000><B100><B110>3715345</B110><B120><B121>CORRECTED EUROPEAN PATENT SPECIFICATION</B121></B120><B130>B8</B130><B132EP>B1</B132EP><B140><date>20240529</date></B140><B150><B151>W1</B151><B153>73</B153><B155><B1551>de</B1551><B1552>Bibliographie</B1552><B1551>en</B1551><B1552>Bibliography</B1552><B1551>fr</B1551><B1552>Bibliographie</B1552></B155></B150><B190>EP</B190></B100><B200><B210>20153723.0</B210><B220><date>20130725</date></B220><B240><B241><date>20210510</date></B241><B242><date>20221205</date></B242></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>201261675663 P</B310><B320><date>20120725</date></B320><B330><ctry>US</ctry></B330><B310>201261680099 P</B310><B320><date>20120806</date></B320><B330><ctry>US</ctry></B330><B310>201261729294 P</B310><B320><date>20121121</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>20240529</date><bnum>202422</bnum></B405><B430><date>20200930</date><bnum>202040</bnum></B430><B450><date>20240410</date><bnum>202415</bnum></B450><B452EP><date>20231020</date></B452EP><B480><date>20240529</date><bnum>202422</bnum></B480></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 405/06        20060101AFI20201002BHEP        </text></classification-ipcr></B510EP><B520EP><classifications-cpc><classification-cpc sequence="1"><text>C07D 405/06        20130101 LI20140123BHEP        </text></classification-cpc><classification-cpc sequence="2"><text>C07D 407/06        20130101 FI20151128BHEP        </text></classification-cpc><classification-cpc sequence="3"><text>A61P  27/02        20180101 LI20200324BHEP        </text></classification-cpc><classification-cpc sequence="4"><text>A61P  29/00        20180101 LI20200324BHEP        </text></classification-cpc><classification-cpc sequence="5"><text>A61P  37/02        20180101 LI20200331BHEP        </text></classification-cpc><classification-cpc sequence="6"><text>A61P  43/00        20180101 LI20200331BHEP        </text></classification-cpc></classifications-cpc></B520EP><B540><B541>de</B541><B542>HERSTELLUNG EINES LFA-1-HEMMERS</B542><B541>en</B541><B542>PREPARATION OF LFA-1 INHIBITOR</B542><B541>fr</B541><B542>PROCÉDÉ DE PRÉPARATION D'UN INHIBITEUR DE LFA-1</B542></B540><B560><B561><text>US-A1- 2011 092 707</text></B561><B562><text>R. Alan Jones: "Quaternary Ammonium Salts: Their Use in Phase-Transfer Catalysis", 2001, Academic Press, London, XP009187190, ISBN: 0-12-389171-X pages 391-411, * page 400 *</text></B562><B562><text>ABDEL-MAGID AHMED F ET AL: "Hydrolysis of polypeptide esters with tetrabutylammonium hydroxide", TETRAHEDRON LETTERS, vol. 39, no. 21, 1998, pages 3391-3394, XP029171361, ISSN: 0040-4039, DOI: 10.1016/S0040-4039(98)00511-5</text></B562></B560></B500><B600><B620><parent><pdoc><dnum><anum>13823367.1</anum><pnum>2877465</pnum></dnum><date>20130725</date></pdoc></parent></B620><B620EP><parent><cdoc><dnum><anum>24169178.1</anum></dnum><date>20240409</date></cdoc></parent></B620EP></B600><B700><B720><B721><snm>ZELLER, James, Robert</snm><adr><str>9113 N 116th Way</str><city>Scottsdale, AZ 85259</city><ctry>US</ctry></adr></B721><B721><snm>VENKATRAMAN, Sripathy</snm><adr><str>111 Van Bael Drive</str><city>Slingerlands, NY 12149</city><ctry>US</ctry></adr></B721><B721><snm>BROT, Elisabeth, C.A.</snm><adr><str>6211 Johnston Road</str><city>Albany, NY 12203</city><ctry>US</ctry></adr></B721><B721><snm>IYER, Subashree</snm><adr><str>1461 Siver Road</str><city>Guilderland, NY 12084</city><ctry>US</ctry></adr></B721><B721><snm>HALL, Michael</snm><adr><str>155 Rosemont Street</str><city>Albany, NY 12206</city><ctry>US</ctry></adr></B721></B720><B730><B731><snm>Bausch + Lomb Ireland Limited</snm><iid>102026142</iid><irf>P077382EP</irf><adr><str>Citywest Business Campus 
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