(19)
(11) EP 3 724 166 A1

(12)

(43) Date of publication:
21.10.2020 Bulletin 2020/43

(21) Application number: 18829243.7

(22) Date of filing: 11.12.2018
(51) International Patent Classification (IPC): 
C07D 223/04(2006.01)
(86) International application number:
PCT/EP2018/084367
(87) International publication number:
WO 2019/115531 (20.06.2019 Gazette 2019/25)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 12.12.2017 EP 17206574
09.05.2018 EP 18171625

(71) Applicant: DSM IP Assets B.V.
6411 TE Heerlen (NL)

(72) Inventors:
  • GEOTTI-BIANCHINI, Piero
    3007 Bern (CH)
  • GYERGYÓI, Katalin
    1066 Budapest (HU)
  • HEIDL, Marc-Matthias
    4303 Kaiseraugst (CH)
  • SZABÓ, András
    1182 Budapest (HU)
  • SZÜCSNÉ CSERÉPI, Stefánia
    1204 Budapest (HU)

   


(54) PROCESS FOR THE MANUFACTURE OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS