(19)
(11) EP 4 118 084 A1

(12)

(43) Date of publication:
18.01.2023 Bulletin 2023/03

(21) Application number: 21715435.0

(22) Date of filing: 11.03.2021
(51) International Patent Classification (IPC): 
C07D 487/04(2006.01)
A61K 31/53(2006.01)
A61P 35/00(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 487/04; A61P 35/00
(86) International application number:
PCT/US2021/021809
(87) International publication number:
WO 2021/183709 (16.09.2021 Gazette 2021/37)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 11.03.2020 IN 202011010365
11.12.2020 IN 202011053964

(71) Applicant: Teva Czech Industries s.r.o.
747 70 Opava-Komarov (CZ)

(72) Inventors:
  • MUTHUSAMY, Anantha Rajmohan
    Sivakasi, Tamilnadu 626189 (IN)
  • SINGH, Amit
    Noida, Uttar Pradesh 201310 (IN)
  • KANNIAH, Sundara Lakshmi
    Vellore, Tamil Nadu 632001 (IN)
  • DAUND, Vaibhav Suresh
    Nasik, Maharashtra 422101 (IN)
  • LUTHRA, Parven Kumar
    Noida, Uttar Pradesh 201304 (IN)
  • WAGH, Yogesh Dhananjay
    Thane, Maharashtra 421503 (IN)
  • SOMASUNDARAM, Meenakshi Sundaram
    Tamilnadu 626203 (IN)

(74) Representative: D Young & Co LLP 
120 Holborn
London EC1N 2DY
London EC1N 2DY (GB)

   


(54) SOLID STATE FORMS OF AVAPRITINIB AND PROCESS FOR PREPARATION THEREOF