MORPHIC FORMS OF TRILACICLIB AND METHODS OF MANUFACTURE THEREOF - Patent 4164653

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EP 4 164 653 A1

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(43)	Date of publication:
	19.04.2023 Bulletin 2023/16

(21)	Application number: 21826036.2

(22)	Date of filing: 15.06.2021

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International Patent Classification (IPC):

A61K 31/519^(2006.01)

C07D 487/20^(2006.01)

(52)	Cooperative Patent Classification (CPC):
	C07D 487/22

(86)	International application number:
	PCT/US2021/037462

(87)	International publication number:
	WO 2021/257587 (23.12.2021 Gazette 2021/51)

(84)	Designated Contracting States:
	AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
	Designated Extension States:
	BA ME
	Designated Validation States:
	KH MA MD TN

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Priority:

15.06.2020 US 202063039372 P
13.11.2020 US 202017097854
27.04.2021 US 202163180578 P

(71)	Applicant: G1 Therapeutics, Inc.
	Research Triangle Park, NC 27709 (US)

(72)	Inventors:
	SCHNEIDER, Stephen Research Triangle Park, NC 27709 (US) SMITH, Alexander Research Triangle Park, NC 27709 (US) WHITE, Hannah, S. Research Triangle Park, NC 27709 (US) STRUM, Jay, Copeland Hillsborough, NC 27278 (US) MAZUREK, Jaroslaw B9030 Mariakerke (BE) WU, Sara Research Triangle Park, NC 27709 (US)

(74)	Representative: Carpmaels & Ransford LLP
	One Southampton Row London WC1B 5HA London WC1B 5HA (GB)

(54)	MORPHIC FORMS OF TRILACICLIB AND METHODS OF MANUFACTURE THEREOF