(19)
(11) EP 4 229 043 A1

(12)

(43) Date of publication:
23.08.2023 Bulletin 2023/34

(21) Application number: 21881315.2

(22) Date of filing: 14.10.2021
(51) International Patent Classification (IPC): 
C07D 261/06(2006.01)
A61K 31/445(2006.01)
C07D 209/04(2006.01)
C07D 261/02(2006.01)
A61K 31/404(2006.01)
C07D 209/02(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 413/14
(86) International application number:
PCT/US2021/071862
(87) International publication number:
WO 2022/082197 (21.04.2022 Gazette 2022/16)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 15.10.2020 US 202063092423 P

(71) Applicant: Eli Lilly and Company
Indianapolis, IN 46285 (US)

(72) Inventors:
  • SWEETANA, Stephanie Ann
    Indianapolis, Indiana 46285 (US)
  • SPROULL, Steven Jerald
    Indianapolis, Indiana 46285 (US)
  • OWENS, Paul K.
    Indianapolis, Indiana 46285 (US)

(74) Representative: Cooley (UK) LLP 
22 Bishopsgate
London EC2N 4BQ
London EC2N 4BQ (GB)

   


(54) POLYMORPHS OF AN FXR AGONIST