(19)
(11) EP 4 271 377 A1

(12)

(43) Date of publication:
08.11.2023 Bulletin 2023/45

(21) Application number: 21916609.7

(22) Date of filing: 29.12.2021
(51) International Patent Classification (IPC): 
A61K 31/42(2006.01)
A61K 31/4245(2006.01)
C07D 261/02(2006.01)
A61K 31/422(2006.01)
A61K 31/41(2006.01)
A61K 31/445(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 413/14; C07D 451/06; C07D 417/14; A61P 43/00
(86) International application number:
PCT/US2021/073153
(87) International publication number:
WO 2022/147448 (07.07.2022 Gazette 2022/27)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 30.12.2020 US 202063132363 P

(71) Applicant: Terns Pharmaceuticals, Inc.
Foster City, California 94404 (US)

(72) Inventors:
  • XU, Yingzi
    Foster City, CA 94404 (US)
  • KLUCHER, Kevin
    Foster City, CA 94404 (US)
  • ROMERO, F., Anthony
    Foster City, CA 94404 (US)

(74) Representative: Cooley (UK) LLP 
22 Bishopsgate
London EC2N 4BQ
London EC2N 4BQ (GB)

   


(54) COMPOUNDS AND METHODS FOR MODULATING FXR