(19)
(11) EP 4 288 427 A1

(12)

(43) Date of publication:
13.12.2023 Bulletin 2023/50

(21) Application number: 22708396.1

(22) Date of filing: 02.02.2022
(51) International Patent Classification (IPC): 
C07D 405/06(2006.01)
C07D 413/06(2006.01)
C07D 409/14(2006.01)
C07D 249/06(2006.01)
C07D 405/12(2006.01)
C07D 401/06(2006.01)
C07D 487/10(2006.01)
C07D 471/14(2006.01)
C07D 405/04(2006.01)
C07D 413/14(2006.01)
C07D 453/02(2006.01)
C07D 401/14(2006.01)
C07D 413/12(2006.01)
C07D 409/06(2006.01)
C07D 405/14(2006.01)
C07D 491/107(2006.01)
C07D 401/12(2006.01)
C07D 471/10(2006.01)
C07D 403/06(2006.01)
C07D 471/04(2006.01)
C07D 487/08(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 405/06; C07D 401/14; C07D 413/06; C07D 413/12; C07D 409/14; C07D 409/06; C07D 249/06; C07D 405/14; C07D 405/12; C07D 491/107; C07D 401/06; C07D 401/12; C07D 487/10; C07D 471/10; C07D 417/14; C07D 403/06; C07D 405/04; C07D 471/04; C07D 413/14; C07D 487/08; C07D 453/02; C07D 471/08; C07D 491/056; C07D 491/048; A61P 25/00; A61P 31/12; A61P 35/00; A61P 37/00
(86) International application number:
PCT/EP2022/052419
(87) International publication number:
WO 2022/167457 (11.08.2022 Gazette 2022/32)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 02.02.2021 US 202163144720 P

(71) Applicant: Liminal Biosciences Limited
Cambridge CB22 3EG (GB)

(72) Inventors:
  • ABBOTT, Shaun
    Cambridge CB22 3EG (GB)
  • DELESELEUC, Mylène
    Cambridge CB22 3EG (GB)
  • MARTEL, Julien
    Cambridge CB22 3EG (GB)
  • BOURQUE, Elyse
    Cambridge CB22 3EG (GB)
  • GREEN, Jeremy
    Cambridge CB22 3EG (GB)
  • LARIVÉE, Alexandre
    Cambridge CB22 3EG (GB)
  • GIGUÈRE, Jean-benoît
    Cambridge CB22 3EG (GB)
  • LANDAGARAY, Elodie
    Cambridge CB22 3EG (GB)
  • STURINO, Claudio
    Cambridge CB22 3EG (GB)
  • NASSER, Nadia Michel
    Cambridge CB22 3EG (GB)

(74) Representative: Petty, Catrin Helen 
Venner Shipley LLP 200 Aldersgate
London EC1A 4HD
London EC1A 4HD (GB)

   


(54) GPR84 ANTAGONISTS AND USES THEREOF