(19)
(11) EP 4 384 493 A1

(12)

(43) Date of publication:
19.06.2024 Bulletin 2024/25

(21) Application number: 22855428.3

(22) Date of filing: 09.08.2022
(51) International Patent Classification (IPC): 
C07C 211/44(2006.01)
C07D 231/00(2006.01)
A61K 31/136(2006.01)
A61P 25/00(2006.01)
A61P 25/16(2006.01)
C07D 213/00(2006.01)
C07D 263/00(2006.01)
A61K 31/395(2006.01)
A61P 25/14(2006.01)
(52) Cooperative Patent Classification (CPC):
A61P 25/14; A61P 25/16; A61P 25/00; C07D 265/30; C07D 241/04; C07D 295/13; C07D 295/135; C07D 401/04; C07D 211/58; C07D 401/12; C07D 405/12; C07D 401/14; C07D 403/12; C07D 211/76; C07D 211/56; C07D 211/96; C07D 211/26; C07D 401/06; C07D 211/18; C07D 211/14; C07D 211/22; C07D 211/48; C07D 211/46; C07D 405/14; C07D 451/04; C07D 487/08; C07D 231/12; C07D 231/38; C07D 213/74; C07D 207/14; C07D 309/14; C07D 207/27; C07D 207/277; C07D 207/273; C07D 205/04; C07D 233/32; C07D 207/08; C07D 215/38; C07D 309/04; C07D 307/79; C07D 277/60; C07D 413/04; C07D 413/14; C07D 417/04; C07D 233/64; C07D 233/61; C07D 239/22; C07D 335/02; C07D 239/47; C07D 209/08; C07D 267/10; C07D 498/08; C07D 491/107; C07D 491/048; C07F 7/0816; C07C 2601/14; C07C 211/53; C07C 217/52; C07C 237/24; C07C 217/08; C07C 2601/08; C07C 2601/04; C07C 2601/18; C07C 215/42; C07C 2603/74; C07C 2602/08; C07C 2602/10; C07C 217/84; C07C 215/44; C07C 2601/02; C07C 211/48; C07C 229/48; C07C 2602/50; C07C 215/10; C07C 217/90; C07C 275/14; C07C 275/26; C07C 307/08; C07C 2602/22; C07C 215/16; C07C 211/51
(86) International application number:
PCT/CN2022/111129
(87) International publication number:
WO 2023/016447 (16.02.2023 Gazette 2023/07)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA ME
Designated Validation States:
KH MA MD TN

(30) Priority: 09.08.2021 WO PCT/CN2021/111481

(71) Applicant: Sironax Ltd
Grand Cayman, KY1-1104 (KY)

(72) Inventors:
  • HOU, Weijie
    Beijing 102206 (CN)
  • ZHANG, Zhiyuan
    Beijing 102206 (CN)
  • XU, Yanping
    Beijing 102206 (CN)
  • JIANG, Yimin
    Beijing 102206 (CN)
  • XU, Xingyu
    Beijing 102206 (CN)
  • HAN, Jianguang
    Beijing 102206 (CN)

(74) Representative: Finnegan Europe LLP 
1 London Bridge
London SE1 9BG
London SE1 9BG (GB)

   


(54) FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF