(19)
(11) EP 4 577 535 A1

(12)

(43) Date of publication:
02.07.2025 Bulletin 2025/27

(21) Application number: 23856487.6

(22) Date of filing: 10.08.2023
(51) International Patent Classification (IPC): 
C07D 401/14(2006.01)
A61K 31/506(2006.01)
C07D 413/14(2006.01)
A61P 35/00(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 413/14; A61P 35/00; C07D 403/14; C07D 405/14
(86) International application number:
PCT/CN2023/112361
(87) International publication number:
WO 2024/041397 (29.02.2024 Gazette 2024/09)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA
Designated Validation States:
KH MA MD TN

(30) Priority: 22.08.2022 WO PCT/CN2022/113873

(71) Applicant: Hangzhou Highlightll Pharmaceutical Co., Ltd.
Hangzhou, Zhejiang 310018 (CN)

(72) Inventors:
  • LIANG, Congxin
    Hangzhou, Zhejiang 310012 (CN)
  • LI, Shuangjiang
    Hangzhou, Zhejiang 310018 (CN)
  • TANG, Xiaojing
    Hangzhou, Zhejiang 310023 (CN)
  • HUANG, Junmin
    Linden (US)

(74) Representative: Dehns 
10 Old Bailey
London EC4M 7NG
London EC4M 7NG (GB)

   


(54) JAK1/JAK2/TYK2 INHIBITORS FOR TOPICAL TREATMENT OF DERMATOLOGICAL DISEASES