(19)
(11) EP 4 583 867 A2

(12)

(88) Date of publication A3:
18.04.2024

(43) Date of publication:
16.07.2025 Bulletin 2025/29

(21) Application number: 23863823.3

(22) Date of filing: 08.09.2023
(51) International Patent Classification (IPC): 
A61K 31/395(2006.01)
A61K 31/44(2006.01)
A61K 31/4995(2006.01)
A61K 31/166(2006.01)
A61K 31/167(2006.01)
A61K 31/33(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 401/14; C07D 401/12; C07D 213/81; C07D 405/14; C07D 401/04; C07D 237/24; C07D 213/82; C07D 513/14; C07D 213/75; C07D 213/66
(86) International application number:
PCT/US2023/032280
(87) International publication number:
WO 2024/054622 (14.03.2024 Gazette 2024/11)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA
Designated Validation States:
KH MA MD TN

(30) Priority: 09.09.2022 US 202263405094 P
09.09.2022 US 202263405096 P
09.09.2022 US 202263405120 P
09.09.2022 US 202263405151 P

(71) Applicant: Latigo Biotherapeutics, Inc.
Thousand Oaks, CA 91320 (US)

(72) Inventors:
  • BAJJI, Ashok
    Thousand Oaks, CA 91320 (US)
  • KAUFMAN, Michael, D.
    Thousand Oaks, CA 91361 (US)
  • BALKOVEC, James, Michael
    Martinsville, NJ 08836 (US)

(74) Representative: HGF 
HGF Limited 1 City Walk
Leeds LS11 9DX
Leeds LS11 9DX (GB)

   


(54) SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE