(19)
(11) EP 4 583 976 A1

(12)

(43) Date of publication:
16.07.2025 Bulletin 2025/29

(21) Application number: 23767907.1

(22) Date of filing: 08.09.2023
(51) International Patent Classification (IPC): 
A61P 35/00(2006.01)
C07D 519/00(2006.01)
A61P 37/00(2006.01)
A61K 31/4353(2006.01)
(52) Cooperative Patent Classification (CPC):
C07D 519/00; A61P 35/00; A61P 37/00
(86) International application number:
PCT/EP2023/074692
(87) International publication number:
WO 2024/052513 (14.03.2024 Gazette 2024/11)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA
Designated Validation States:
KH MA MD TN

(30) Priority: 09.09.2022 EP 22194841

(71) Applicant: Chiesi Farmaceutici S.p.A.
43122 Parma (IT)

(72) Inventors:
  • ACCETTA, Alessandro
    43122 Parma (IT)
  • CUZZOLIN, Alberto
    43122 Parma (IT)
  • RANCATI, Fabio
    43122 Parma (IT)
  • RIZZI, Andrea
    43122 Parma (IT)
  • ELENKOV, Ivaylo Jivkov
    43122 Parma (IT)
  • MESI , Milan
    43122 Parma (IT)
  • FIORELLI, Claudio
    43122 Parma (IT)

(74) Representative: Chiesi Farmaceutici S.p.A. 
Via Palermo, 26/A
43122 Parma
43122 Parma (IT)

   


(54) HETEROCYCLIC DERIVATIVES AS JANUS KINASE INHIBITORS