(19)
(11) EP 4 770 661 A2

(12)

(88) Date of publication A3:
17.04.2025

(43) Date of publication:
08.07.2026 Bulletin 2026/28

(21) Application number: 24861224.4

(22) Date of filing: 30.08.2024
(51) International Patent Classification (IPC): 
A61K 38/19(2006.01)
A61K 38/16(2006.01)
(52) Cooperative Patent Classification (CPC):
A61P 35/00; A61K 45/06; A61K 31/675; A61K 31/395; A61K 38/193; A61K 38/08; A61K 38/12
 
C-Sets:
  1. A61K 38/12, A61K 2300/00;
  2. A61K 31/675, A61K 2300/00;
  3. A61K 31/395, A61K 2300/00;
  4. A61K 38/193, A61K 2300/00;
  5. A61K 38/08, A61K 2300/00;

(86) International application number:
PCT/US2024/044862
(87) International publication number:
WO 2025/050038 (06.03.2025 Gazette 2025/10)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA
Designated Validation States:
GE KH MA MD TN

(30) Priority: 30.08.2023 US 202363579773 P

(71) Applicants:
  • GPCR Therapeutics, Inc.
    Seoul 08790, (KR)
  • Cardarelli, Josephine
    San Carlos, California 94070 (US)

(72) Inventors:
  • SUKHTANKAR, Devki
    Fremont, California 94555 (US)
  • CAYTON, Thomas
    Pleasanton, California 94566 (US)
  • CARDARELLI, Josephine
    San Carlos, California 94070 (US)

(74) Representative: Berggren Oy 
P.O. Box 16 Fabianinkatu 21
00101 Helsinki
00101 Helsinki (FI)

   


(54) GPCR INHIBITORS AND USES THEREOF