(19)
(11) EP 4 798 588 A1

(12)

(43) Date of publication:
02.09.2026 Bulletin 2026/36

(21) Application number: 24881884.1

(22) Date of filing: 24.10.2024
(51) International Patent Classification (IPC): 
C07D 471/04(2006.01)
A61K 31/437(2006.01)
C07D 209/10(2006.01)
C07D 409/06(2006.01)
A61K 31/444(2006.01)
A61P 35/00(2006.01)
C07D 231/56(2006.01)
(52) Cooperative Patent Classification (CPC):
A61P 35/00; C07D 209/10; C07D 231/56; C07D 409/06; C07D 471/04; C07D 519/00
(86) International application number:
PCT/IB2024/060467
(87) International publication number:
WO 2025/088534 (01.05.2025 Gazette 2025/18)
(84) Designated Contracting States:
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC ME MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated Extension States:
BA
Designated Validation States:
GE KH MA MD TN

(30) Priority: 27.10.2023 KR 20230145969

(71) Applicant: Dong-A ST Co., Ltd.
Dongdaemun-gu Seoul 02587 (KR)

(72) Inventors:
  • CHOI, Sunho
    Seoul 06732 (KR)
  • KONG, Younggyu
    Yongin-si, Gyeonggi-do 17066 (KR)
  • KIM, Yoonjung
    Suwon-si, Gyeonggi-do 16519 (KR)
  • PARK, Youngjun
    Yongin-si, Gyeonggi-do 17046 (KR)
  • PARK, Jihyun
    Yongin-si, Gyeonggi-do 17073 (KR)
  • BAEK, Gyerim
    Yongin-si, Gyeonggi-do 17081 (KR)
  • SOH, Hyeyeon
    Yongin-si, Gyeonggi-do 16846 (KR)
  • YOO, Jaewook
    Yongin-si, Gyeonggi-do 17066 (KR)
  • LEE, Okyoung
    Hwaseong-si, Gyeonggi-do 18496 (KR)
  • JEONG, Youngmin
    Seoul 05764 (KR)
  • JUNG, Hyeonseok
    Yongin-si, Gyeonggi-do 17067 (KR)
  • HAN, Taedong
    Yongin-si, Gyeonggi-do 17080 (KR)

(74) Representative: HGF 
HGF Limited 4th Floor, 1 City Square
Leeds LS1 2ES
Leeds LS1 2ES (GB)

   


(54) BICYCLIC HETEROCYCLE COMPOUNDS AS TEAD INHIBITOR